Related drugs targeting FXR
FXR agonists | Alias | Molecular formula | Chemical structure | R & D stage | References |
---|---|---|---|---|---|
Obeticholic acid | 6-Ethyl-chenodeoxycholic-acid, OCA | C26H44O4 | ![]() | Approval to market | [24, 25] |
GW4064 | GW-4064 | C28H22Cl3NO4 | ![]() | Preclinical | [24, 25] |
Cilofexor | CILO, GS-9674 | C32H33Cl3N4O8 | ![]() | Phase III | [24, 25] |
Tropifexor | LJN-452, NVP-LJN452-NXA | C29H25F4N3O5S | ![]() | Phase II | [24, 25] |
EDP-305 | EDP 305 | C36H58N2O5S | ![]() | Phase II | [27] |
LY-2562175 | None | C28H27Cl2N3O4 | ![]() | Phase II | [24, 25] |