The primary amino acid sequences of Ala scan peptides were listed with the inhibition rate at a fixed concentration of 1 μM. Those with > 90% inhibition were further characterized for IC50
Name | Amino acid sequence | Inhibition (%) | IC50 ± SD (nM) |
---|---|---|---|
BCP-8B | Ala-Cys-Ala-Gly-Arg-Cys-Pro-Ser-Ala-Cys-Leu | 93.8% | 153.63 ± 17.87 nM |
BCP-9B | Ala-Cys-Ala- | 66.2% | - |
BCP-10B | Ala-Cys-Ala-Gly- | 46.6% | - |
BCP-11B | Ala-Cys-Ala-Gly-Arg-Cys- | 81.8% | - |
BCP-12B | Ala-Cys-Ala-Gly-Arg-Cys-Pro- | 69.7% | - |
BCP-13B | Ala-Cys-Ala-Gly-Arg-Cys-Pro-Ser-Ala-Cys- | 3.4% | - |
BCP-14B | Ala-Cys- | 10.4% | - |
BCP-15B | Ala-Cys-Ala- | 99.5% | 62.00 ± 7.31 nM |
BCP-16B | Ala-Cys-Ala-Gly-Arg-Cys- | 95.8% | 116.67 ± 7.79 nM |
-: no data. SD: standard deviation; IC50: half-maximal inhibitory concentration